Antibody Drug Conjugates: Linkers and Payloads

Linker Design

Payload Design

Payload Linker Attachment

  • Diverse linker design and synthesis – Cleavable and Non-cleavable
  • Druggability parameters
  • Target Potency
  • Cytotoxicity
  • Overcoming Efflux challenges
  • Permeability
  • IP challenges
  • Design of novel synthesis
  • Establish the attachment site.